Pharmacology is one of the pillars of medicine, bridging biological science and therapeutics. Understanding drug names, their classes, and uses is essential for safe clinical practice, prescription writing, and exam success.
Drug lists often look overwhelming—but when organized alphabetically with pharmacological classes and uses, they become a powerful learning resource. This article provides a complete drug reference list (A → Z) designed for students, healthcare professionals, and exam aspirants.
A → Z Drug Names with Pharmacology Reference
A Drugs
Drug | Class | Uses | Clinical Notes |
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Abacavir | Antiretroviral (NRTI) | HIV/AIDS treatment | Used in HAART regimen. |
Acetaminophen (Paracetamol) | Analgesic, Antipyretic | Pain, fever | Overdose causes hepatotoxicity. |
Acetylcysteine | Mucolytic, Antidote | COPD (mucus thinning), paracetamol overdose | Restores glutathione. |
Acyclovir | Antiviral | Herpes simplex, Varicella zoster | Safe in pregnancy. |
Albuterol (Salbutamol) | Beta-2 agonist | Asthma, COPD | Inhaler for bronchospasm relief. |
Alteplase (tPA) | Thrombolytic | Acute MI, ischemic stroke | Bleeding risk. |
Aluminum Hydroxide | Antacid | GERD, peptic ulcer | Can cause constipation. |
B Drugs
Drug | Class | Uses | Clinical Notes |
---|
Bisacodyl | Laxative | Constipation relief | Stimulates bowel movement. |
Bumetanide | Loop diuretic | Edema, CHF | Stronger than furosemide. |
Bupropion | Atypical antidepressant | Depression, smoking cessation | Lowers seizure threshold. |
Buspirone | Anxiolytic (5-HT1A partial agonist) | Generalized anxiety disorder | Non-sedating. |
C Drugs
Drug | Class | Uses | Clinical Notes |
---|
Calcium Carbonate | Antacid, supplement | Hypocalcemia, osteoporosis | May cause constipation. |
Carbamazepine | Anticonvulsant | Epilepsy, trigeminal neuralgia | Risk of agranulocytosis. |
Captopril | ACE inhibitor | Hypertension, CHF | Can cause dry cough, hyperkalemia. |
Cephalosporins | Antibiotic | Bacterial infections | Classified into generations. |
Chlorpromazine | Antipsychotic (typical) | Schizophrenia, mania | Causes sedation, EPS. |
Cimetidine | H2 blocker | GERD, peptic ulcer | Inhibits CYP450. |
Ciprofloxacin | Fluoroquinolone antibiotic | UTI, GI infections | Contraindicated in children. |
D Drugs
Drug | Class | Uses | Clinical Notes |
---|
Diazepam | Benzodiazepine | Anxiety, seizures, muscle relaxant | Risk of dependence. |
Digoxin | Cardiac glycoside | CHF, atrial fibrillation | Toxicity causes arrhythmias. |
Diphenhydramine | Antihistamine (1st gen) | Allergy, motion sickness | Causes sedation. |
Doxycycline | Tetracycline antibiotic | Rickettsia, Chlamydia | Avoid in children & pregnancy. |
E Drugs
Drug | Class | Uses | Clinical Notes |
---|
Enalapril | ACE inhibitor | Hypertension, CHF | Risk of hyperkalemia. |
Enoxaparin | Low molecular weight heparin | DVT, PE prevention | Safer than unfractionated heparin. |
Epinephrine | Catecholamine | Anaphylaxis, cardiac arrest | First-line in anaphylaxis. |
Erythromycin | Macrolide antibiotic | Respiratory infections | CYP3A4 inhibitor. |
F Drugs
Drug | Class | Uses | Clinical Notes |
---|
Fentanyl | Opioid analgesic | Severe pain, anesthesia | Very potent, risk of respiratory depression. |
Fluconazole | Antifungal | Candidiasis, cryptococcosis | Inhibits CYP450. |
Fluoxetine | SSRI antidepressant | Depression, OCD | Long half-life. |
Furosemide | Loop diuretic | Pulmonary edema, hypertension | Causes hypokalemia. |
G Drugs
Drug | Class | Uses | Clinical Notes |
---|
Gabapentin | Anticonvulsant / Neuropathic pain agent | Epilepsy, neuropathic pain, fibromyalgia | Causes sedation, dizziness. |
Gentamicin | Aminoglycoside antibiotic | Severe Gram-negative infections | Nephrotoxic, ototoxic. |
Glucagon | Hormone (pancreatic) | Severe hypoglycemia, beta-blocker overdose | Raises blood glucose quickly. |
Guaifenesin | Expectorant | Cough with mucus | Common in OTC cough syrups. |
H Drugs
Drug | Class | Uses | Clinical Notes |
---|
Haloperidol | Typical antipsychotic | Schizophrenia, acute psychosis, Tourette’s | Causes extrapyramidal symptoms (EPS). |
Heparin | Anticoagulant | DVT, PE, MI | Antidote = Protamine sulfate. |
Hydrochlorothiazide | Thiazide diuretic | Hypertension, CHF | Risk of hypokalemia. |
Hydrocodone | Opioid analgesic | Moderate to severe pain | High abuse potential. |
I Drugs
Drug | Class | Uses | Clinical Notes |
---|
Ibuprofen | NSAID | Pain, fever, inflammation | Risk of GI irritation. |
Iloperidone | Atypical antipsychotic | Schizophrenia | Fewer EPS than typical antipsychotics. |
Imipenem | Carbapenem antibiotic | Broad-spectrum bacterial infections | Resistant to most β-lactamases. |
Imipramine | Tricyclic antidepressant (TCA) | Depression, enuresis | Anticholinergic side effects. |
Insulin | Hormone | Diabetes mellitus | Risk of hypoglycemia. |
Ipratropium | Anticholinergic bronchodilator | Asthma, COPD | Inhaler, slower than albuterol. |
Irbesartan | ARB (angiotensin receptor blocker) | Hypertension | Alternative to ACE inhibitors. |
K Drugs
Drug | Class | Uses | Clinical Notes |
---|
Ketoconazole | Antifungal | Fungal infections, Cushing’s syndrome (off-label) | Inhibits CYP450. |
L Drugs
Drug | Class | Uses | Clinical Notes |
---|
Lactulose | Osmotic laxative | Hepatic encephalopathy, constipation | Reduces ammonia absorption. |
Lamivudine | Antiretroviral (NRTI) | HIV, Hepatitis B | Used in HAART. |
Lamotrigine | Anticonvulsant | Epilepsy, bipolar disorder | Risk of Stevens–Johnson syndrome. |
Lansoprazole | Proton pump inhibitor (PPI) | GERD, peptic ulcer | Long-term use → B₁₂ deficiency. |
Levodopa/Carbidopa | Dopamine precursor + decarboxylase inhibitor | Parkinson’s disease | Reduces tremor and rigidity. |
Levothyroxine | Synthetic T₄ hormone | Hypothyroidism | Monitor TSH levels. |
Lisinopril | ACE inhibitor | Hypertension, CHF | Causes cough, hyperkalemia. |
Lithium | Mood stabilizer | Bipolar disorder | Narrow therapeutic index; monitor levels. |
Lorazepam | Benzodiazepine | Anxiety, seizures | Intermediate-acting, safer in liver disease. |
Losartan | ARB | Hypertension | No cough (unlike ACE inhibitors). |
Lovastatin | Statin | Hyperlipidemia | Risk of rhabdomyolysis. |
M Drugs
Drug | Class | Uses | Clinical Notes |
---|
Magnesium Hydroxide | Antacid, laxative | Constipation, heartburn | Can cause diarrhea. |
Mannitol | Osmotic diuretic | Raised ICP, acute glaucoma | Risk of electrolyte imbalance. |
Metformin | Biguanide | Type 2 diabetes | Risk of lactic acidosis; weight neutral. |
Methadone | Opioid agonist | Opioid dependence, chronic pain | Long half-life; QT prolongation. |
Methotrexate | Antimetabolite (antifolate) | Cancer, autoimmune diseases (RA, psoriasis) | Teratogenic, hepatotoxic. |
Metoprolol | Beta-1 blocker | Hypertension, angina, CHF | Cardioselective. |
Metronidazole | Antiprotozoal / Antibiotic | Amoebiasis, giardiasis, anaerobic infections | Disulfiram-like reaction with alcohol. |
Morphine | Opioid analgesic | Severe pain, palliative care | Risk of respiratory depression. |
Medical Abbreviations and Acronyms List – Complete Healthcare Reference
N Drugs
Drug | Class | Uses | Clinical Notes |
---|
Naloxone | Opioid antagonist | Opioid overdose | Short half-life, may need repeat doses. |
Naratriptan | Triptan (5-HT₁ agonist) | Migraine | Vasoconstrictive action. |
Nevirapine | Antiretroviral (NNRTI) | HIV treatment | Rash and hepatotoxicity risk. |
Nifedipine | Calcium channel blocker | Hypertension, angina | Causes reflex tachycardia. |
Nitroglycerin | Nitrate | Angina, hypertensive crisis | Sublingual for acute relief. |
Nitroprusside | Vasodilator | Hypertensive emergency | Can cause cyanide toxicity. |
Norepinephrine | Catecholamine | Septic shock, hypotension | Strong alpha-agonist. |
Nortriptyline | TCA | Depression, neuropathic pain | Anticholinergic side effects. |
Nystatin | Antifungal | Oral candidiasis (thrush) | Not absorbed orally. |
O Drugs
Drug | Class | Uses | Clinical Notes |
---|
Olanzapine | Atypical antipsychotic | Schizophrenia, bipolar disorder | Weight gain, metabolic syndrome. |
Omeprazole | PPI | GERD, ulcers | Long-term risk: osteoporosis. |
Ondansetron | 5-HT₃ antagonist | Chemotherapy-induced nausea/vomiting | Can cause QT prolongation. |
Oxybutynin | Anticholinergic | Overactive bladder | Dry mouth, constipation. |
Oxycodone | Opioid analgesic | Moderate to severe pain | High addiction potential. |
Oxytocin | Hormone | Labor induction, postpartum hemorrhage | Risk of uterine rupture if misused. |
P Drugs
Drug | Class | Uses | Clinical Notes |
---|
Pantoprazole | PPI | GERD, Zollinger–Ellison syndrome | Safer with fewer interactions. |
Paroxetine | SSRI | Depression, anxiety disorders | Causes sexual dysfunction. |
Penicillin | Beta-lactam antibiotic | Streptococcal infections, syphilis | Allergic reactions common. |
Phenelzine | MAOI | Depression (refractory) | Hypertensive crisis with tyramine foods. |
Phenobarbital | Barbiturate | Epilepsy, sedation | Risk of dependence, respiratory depression. |
Prednisone | Corticosteroid | Inflammation, asthma, autoimmune | Long-term use: Cushingoid features. |
Propranolol | Non-selective beta blocker | Hypertension, arrhythmia, anxiety | Contraindicated in asthma. |
Progesterone | Hormone | Contraception, HRT | Can cause mood changes. |
R Drugs
Drug | Class | Uses | Clinical Notes |
---|
Ranitidine | H₂ blocker | Peptic ulcer, GERD | Withdrawn in many markets (NDMA impurity). |
Rifampin | Antitubercular | TB treatment | Turns body fluids orange. |
Risperidone | Atypical antipsychotic | Schizophrenia, bipolar disorder | Can cause hyperprolactinemia. |
Rosuvastatin | Statin | Hyperlipidemia | Stronger LDL lowering. |
S Drugs
Drug | Class | Uses | Clinical Notes |
---|
Sertraline | SSRI | Depression, PTSD, OCD | Fewer drug interactions. |
Sildenafil | PDE-5 inhibitor | Erectile dysfunction, pulmonary hypertension | Contraindicated with nitrates. |
Simvastatin | Statin | Hypercholesterolemia | Risk of muscle toxicity. |
Spironolactone | Potassium-sparing diuretic, aldosterone antagonist | CHF, cirrhosis, PCOS | Causes gynecomastia. |
Sumatriptan | Triptan | Acute migraine | Vasoconstriction risk. |
T Drugs
Drug | Class | Uses | Clinical Notes |
---|
Temazepam | Benzodiazepine | Insomnia | Short-acting. |
Terbutaline | Beta-2 agonist | Asthma, preterm labor | Causes tachycardia, tremors. |
Testosterone | Androgen hormone | Hypogonadism, delayed puberty | Risk of prostate cancer. |
Theophylline | Bronchodilator (methylxanthine) | Asthma, COPD | Narrow therapeutic index. |
Torsemide | Loop diuretic | Edema, hypertension | Similar to furosemide. |
Trazodone | Antidepressant (SARI) | Depression, insomnia | Causes priapism (rare). |
Trimethoprim | Antimicrobial | UTI | Often combined with sulfamethoxazole. |
V Drugs
Drug | Class | Uses | Clinical Notes |
---|
Valproic Acid | Anticonvulsant, mood stabilizer | Epilepsy, bipolar disorder | Teratogenic (neural tube defects). |
Vancomycin | Glycopeptide antibiotic | MRSA, C. difficile (oral) | Risk of “Red Man syndrome.” |
Varenicline | Nicotinic receptor partial agonist | Smoking cessation | Risk of vivid dreams, depression. |
Vilazodone | SSRI + 5-HT1A agonist | Depression | Less sexual dysfunction. |
W, X, Y, Z Drugs
Drug | Class | Uses | Clinical Notes |
---|
Warfarin | Vitamin K antagonist | Anticoagulant (AF, DVT, PE) | Requires INR monitoring. |
Zafirlukast | Leukotriene receptor antagonist | Asthma maintenance | Can cause liver toxicity. |
FAQs
Q1. What are the most important drugs to memorize for exams?
Analgesics, antibiotics, antidiabetics, antihypertensives, and psychotropic drugs are high-yield.
Q2. How can I quickly learn drug names and classes?
Using mnemonics, flashcards, and grouping drugs by suffixes (-pril, -olol, -azole).
Q3. Why do many drugs have similar names?
Because suffixes often denote drug class (e.g., “-azole” for antifungals).
Q4. What is the difference between generic and brand names?
Generic = chemical/standard name (e.g., Paracetamol). Brand = trade name (e.g., Crocin, Tylenol).
Q5. Which drugs are on the WHO Essential Medicines List?
Paracetamol, Amoxicillin, Insulin, Omeprazole, Morphine, Warfarin, etc.